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Woburn, MA, United States of America

Arqule, Inc.

USPTO Granted Patents = 104

% Expired Patents = 17.3

CIPO Patents = 1

EPO Patents = 22

Trademarks = 2

Forward Citations = 544

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129 inventors (with patents filed for the assignee):

Mark Anthony Ashwell (36 out of 45 patents)

Manish Tandon (24 out of 24 patents)

Jean-Marc Lapierre (23 out of 34 patents)

4. Nivedita Namdev (21 out of 21 patents)

5. Yanbin Liu (18 out of 18 patents)

6. Rocio Palma (17 out of 17 patents)

7. Syed M Ali (17 out of 18 patents)

8. Jason J Hill (17 out of 55 patents)

9. David P Reed (13 out of 13 patents)

10. Joseph C Hogan, Jr (13 out of 13 patents)

11. David S Casebier (12 out of 38 patents)

12. David Vensel (12 out of 12 patents)

13. Craig G Bates (12 out of 15 patents)

14. Sudharshan Eathiraj (11 out of 11 patents)

15. Chiang Jia Li (10 out of 57 patents)

Core Competencies:

Cancer Treatment

Kinase Inhibitors

Heterocyclic Compounds

Amino-Pyrrolopyrimidinone

Substituted Imidazopyridines

Pyrroloquinolinyl-Pyrrolidine

Prodrug Compositions

Triazine Derivatives

104 patents: Sort by Forward Citations

1. 11279679 - Methods for preparing substituted 5,6-dihydro-6-phenylbenzo[f]isoquinolin-2-amine (2022-03-22),

2. 11020400 - Tetrahydropyranyl amino-pyrrolopyrimidinone and methods of use thereof (2021-06-01),

3. 11020398 - Amino-pyrrolopyrimidinone compounds and methods of use thereof (2021-06-01),

4. 10975087 - Solid forms of tetrahydropyranyl amino-pyrrolopyrimidinone compounds (2021-04-13),

5. 10933065 - Tetrahydropyranyl amino-pyrrolopyrimidinone and methods of use thereof (2021-03-02),

6. 10766868 - Methods for preparing substituted 5,6-dihydro-6-phenylbenzo[f]isoquinolin-2-amine (2020-09-08),

7. 10717710 - Solid forms of substituted 5,6-dihydro-6-phenylbenzo[F]isoquinolin-2-amine compounds (2020-07-21),

8. 10245263 - Tetrahydropyranyl amino-pyrrolopyrimidinone and methods of use thereof (2019-04-02),

9. 10227311 - Solid forms of substituted 5,6-dihydro-6-phenylbenzo[F]isoquinolin-2-amine compounds (2019-03-12),

10. 10093632 - Methods for preparing substituted 5,6-dihydro-6-phenylbenzo[F]isoquinolin-2-amine (2018-10-09),

11. 9981921 - Solid forms of substituted 5,6-dihydro-6-phenylbenzo[F]isoquinolin-2-amine compounds (2018-05-29),

12. 9949981 - Compositions and methods for treating proliferation disorders (2018-04-24),

13. 9834556 - Process of preparing 3-(3-(4-aminocyclobutyl)phenyl)-5-phenyl-3H-imidazo[4,5-B]pyridin-2-YL)pyridin-2-amine (2017-12-05),

14. 9834519 - Methods for preparing substituted 5,6-dihydro-6-phenylbenzo[F]isoquinolin-2-amine (2017-12-05),

15. 9642847 - Combinational compositions and methods for treatment of cancer (2017-05-09),

Company Overview

Arqule, Inc., based in Woburn, MA, specializes in the development of innovative pharmaceutical compounds aimed at treating cancer. The company focuses on advanced therapeutic modalities, particularly kinase inhibitors and various heterocyclic compounds. Its research encompasses a range of specialized chemical entities, including amino-pyrrolopyrimidinones and substituted imidazopyridines, contributing to the evolving landscape of targeted cancer therapies. Arqule's commitment to scientific excellence positions it as a key player in the oncology sector.

Profile summary synthesized from public USPTO records and patent filings.

Company Badge

USPTO Data Jan 1 1976 - Oct 13 2026

104 Patents

#2 in Woburn, MA

#197 in Massachusetts

#3,663 in US

#7,525 in the World

Woburn, MA, United States of America

Arqule, Inc.

Forward Citations = 544

129 inventors:

Mark Anthony Ashwell (36 out of 45 patents)

Manish Tandon (24 out of 24 patents)

Jean-Marc Lapierre (23 out of 34 patents)

4. Nivedita Namdev (21 out of 21 patents)

5. Yanbin Liu (18 out of 18 patents)

IDiyas Innovation Intelligence. (2026). Company Patent Portfolio: Arqule, Inc.. Retrieved from https://idiyas.com/company/arqule

Data source: USPTO (United States Patent and Trademark Office) public patent records. Weekly synchronization. How IDiyas builds this profile

Data Sources: USPTO Patent Grant XML, Patent Center, EPO & CIPO • Normalized by IDiyas Innovation Graph. Methodology & provenance architecturePlease report any incorrect information to [email protected]

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