The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Feb. 20, 2024

Filed:

May. 18, 2022
Applicant:

Bracco Suisse SA, Manno, CH;

Inventors:

Federico Maisano, Lodi, IT;

Federico Crivellin, Caselle Torinese, IT;

Thierry Bettinger, Peillonnex, FR;

Philippe Bussat, Pers-Jussy, FR;

Samir Cherkaoui, Feigeres, FR;

Christian Koller, Geneva, CH;

Adrian Lobito, Belmont, CA (US);

Assignee:

Bracco Suisse, Manno, CH;

Attorney:
Primary Examiner:
Int. Cl.
CPC ...
C07K 14/705 (2006.01); A61K 49/00 (2006.01); A61K 49/22 (2006.01); A61K 49/08 (2006.01); C12N 9/10 (2006.01); A61K 38/00 (2006.01);
U.S. Cl.
CPC ...
C07K 14/70564 (2013.01); A61K 49/0032 (2013.01); A61K 49/0056 (2013.01); A61K 49/0084 (2013.01); A61K 49/085 (2013.01); A61K 49/221 (2013.01); A61K 49/223 (2013.01); C07K 14/705 (2013.01); C12N 9/1051 (2013.01); A61K 38/00 (2013.01); C12Y 204/01039 (2013.01); C12Y 204/01068 (2013.01); G01N 2333/70564 (2013.01);
Abstract

The invention discloses a recombinant protein (P-selectin glycoprotein ligand-1 and Neural Retina-specific Leucine Zipper) PSGL-1-NRL chimeric protein comprising a Selectin Binding domain and a non-covalent dimerization domain, which is a leucine zipper and is more preferably the leucine zipper domain of the human or mouse Neural Retina-specific Leucine Zipper. The chimeric protein further comprises a covalent dimerization domain with at least one cysteine suitable to form a disulfide bridge with another chimeric protein to form a homodimer. In the chimeric protein, the PSGL-1 domain corresponds to the extracellular region of Human PSGL-1 and is more preferably the selectin binding region of the mature protein. The chimeric protein is correctly post-translationally modified and is efficiently expressed in a mammalian system. It is sulfated, O-linked glycosylated and sialylated and binds P, E and L selectin, allowing in vivo and in vitro targeting for diagnostic or therapeutic purposes.


Find Patent Forward Citations

Loading…