The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Jun. 06, 2017

Filed:

Jun. 18, 2015
Applicants:

Abbvie B.v., Hoofddorp, NL;

Abbvie Inc., North Chicago, IL (US);

Inventors:

Pieter Smid, Hoofddorp, NL;

Wouter I. Iwema Bakker, Hoofddorp, NL;

Hein K. A. C. Coolen, Hoofddorp, NL;

Leonardus A. J. M. Sliedregt, Hoofddorp, NL;

Maria J. P. van Dongen, Hoofddorp, NL;

Jacobus A. J. den Hartog, Hoofddorp, NL;

Adrian Hobson, Worcester, MA (US);

Assignees:

Abbvie B.V., Hoofddorp, NL;

AbbiVie Inc., North Chicago, IL (US);

Attorney:
Primary Examiner:
Int. Cl.
CPC ...
A01N 43/00 (2006.01); A01N 43/46 (2006.01); A61K 31/55 (2006.01); C07D 491/048 (2006.01); C07D 487/04 (2006.01); C07D 491/04 (2006.01); C07D 498/04 (2006.01); C07D 513/04 (2006.01); C07D 471/04 (2006.01); C07D 495/04 (2006.01);
U.S. Cl.
CPC ...
C07D 491/048 (2013.01); C07D 471/04 (2013.01); C07D 487/04 (2013.01); C07D 491/04 (2013.01); C07D 495/04 (2013.01); C07D 498/04 (2013.01); C07D 513/04 (2013.01);
Abstract

The present invention relates to a fused heterocyclic derivative of the formula (I) The variables R1-R4, z, A, Q, X and Y are as defined in the claims. The following heterocycles are exemplified sub-structures of formula (I): The compounds of formula (I) are modulators of the S1P receptor (Sphingosine-1-phosphate receptor), More specifically, they are agonists of S1P5. The compounds have therapeutic use in treatment of cognitive disorders, age-relate cognitive decline and dementia.


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