The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Feb. 14, 2017

Filed:

Dec. 08, 2011
Applicants:

John Gilmer, Dublin, IE;

Mark Ledwidge, Cork, IE;

Ken Mcdonald, Dublin, IE;

Pat O'flynn, Cork, IE;

Inventors:

John Gilmer, Dublin, IE;

Mark Ledwidge, Cork, IE;

Ken McDonald, Dublin, IE;

Pat O'Flynn, Cork, IE;

Assignee:
Attorneys:
Primary Examiner:
Int. Cl.
CPC ...
A61K 45/06 (2006.01); A61K 47/48 (2006.01); A61K 31/00 (2006.01); A61K 31/21 (2006.01); A61K 31/4458 (2006.01); A61K 31/4462 (2006.01); A61K 31/4465 (2006.01); A61K 31/65 (2006.01); C07C 237/26 (2006.01);
U.S. Cl.
CPC ...
A61K 47/481 (2013.01); A61K 31/00 (2013.01); A61K 31/21 (2013.01); A61K 31/4458 (2013.01); A61K 31/4462 (2013.01); A61K 31/4465 (2013.01); A61K 31/65 (2013.01); A61K 45/06 (2013.01); C07C 237/26 (2013.01);
Abstract

A combination of: a first tetracycline (TC) component; and a second component capable of releasing nitric oxide (NO) or a nitrate capable of mimicking NO effects in vivo (NO mimetic). The combinations of the invention advantageously act as more effective MMP modulators with selective reductions in circulating MMP-9 levels in-vivo and inhibitory effects on MMP-2 and MMP-9 levels in-vitro. The combinations of the invention also advantageously act as modulators of inflammation mediators. The co-existence of abnormalities of MMP enzymes and inflammation in many diseases make these characteristics advantageous. Therefore, the various combinations of the invention find utility in medical applications where MMPs and/or inflammation is implicated.


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