The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Aug. 09, 2022

Filed:

Jun. 10, 2020
Applicant:

Korea Institute of Science and Technology, Seoul, KR;

Inventors:

Gyo Chang Keum, Seoul, KR;

Ashraf Kareem El-Damasy, Seoul, KR;

Hee Won Jin, Seoul, KR;

Taek Kang, Seoul, KR;

Eun Kyoung Bang, Seoul, KR;

Attorney:
Primary Examiner:
Int. Cl.
CPC ...
C07D 413/12 (2006.01); C07D 403/12 (2006.01); C07D 231/56 (2006.01); A61P 35/02 (2006.01);
U.S. Cl.
CPC ...
C07D 413/12 (2013.01); A61P 35/02 (2018.01); C07D 231/56 (2013.01); C07D 403/12 (2013.01);
Abstract

Disclosed are a compound selected from novel indazole derivatives, pharmaceutically acceptable salts thereof, hydrates thereof and stereoisomers thereof, a method for preparing the compound, and a pharmaceutical composition for preventing, alleviating or treating cancer containing the compound as an active ingredient. The novel indazole derivatives exhibit excellent ABL/DDR1 inhibitory efficacy and anti-proliferative efficacy against cancer cells, specifically blood cancer cells, and inhibitory activity against ABL T315I point mutations, thus being useful for the prevention, alleviation or treatment of cancer, specifically blood cancer, especially chronic myelogenous leukemia.


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