The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Oct. 31, 2017

Filed:

Jan. 11, 2008
Applicants:

Francesco Berti, Siena, IT;

Paolo Costantino, Siena, IT;

Alessandro Pianigiani, Siena, IT;

Inventors:

Angela Bardotti, Siena, IT;

Francesco Berti, Siena, IT;

Paolo Costantino, Siena, IT;

Attorney:
Primary Examiner:
Assistant Examiner:
Int. Cl.
CPC ...
C08B 37/00 (2006.01); A61K 39/095 (2006.01); A61K 47/48 (2006.01); C07H 13/00 (2006.01); A61K 39/00 (2006.01);
U.S. Cl.
CPC ...
C08B 37/00 (2013.01); A61K 39/095 (2013.01); A61K 47/4833 (2013.01); C07H 13/00 (2013.01); C08B 37/006 (2013.01); A61K 2039/55505 (2013.01); A61K 2039/6037 (2013.01);
Abstract

Modified capsular saccharides comprising a blocking group at a hydroxyl group position on at least one of the monosaccharide units of the corresponding native capsular saccharide, wherein the blocking group is of the formula (Ia) or (Ib): —OX—Y (Ia) or —O—R(Ib) wherein X is C(O), S(O) or SO; Y is NRRor R; Ris Calkyl substituted with 1, 2 or 3 groups independently selected from hydroxyl, sulphydryl and amine; Ris H or Calkyl; and Ris Calkyl; processes for modifying a capsular saccharide with the blocking groups; saccharide-protein conjugates comprising the modified capsular saccharide; processes for making the saccharide-protein conjugates, pharmaceutical compositions comprising the modified capsular saccharides and/or saccharide-protein conjugates; and methods and uses of the same.


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