The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Jun. 06, 2017

Filed:

Jan. 19, 2011
Applicants:

Steven L. Colletti, Princeton Junction, NJ (US);

Zhengwu James Deng, Eagleville, PA (US);

Matthew G. Stanton, Marlton, NJ (US);

Weimin Wang, Churchville, PA (US);

Ivory Hills, Deerfield, MA (US);

Inventors:

Steven L. Colletti, Princeton Junction, NJ (US);

Zhengwu James Deng, Eagleville, PA (US);

Matthew G. Stanton, Marlton, NJ (US);

Weimin Wang, Churchville, PA (US);

Ivory Hills, Deerfield, MA (US);

Assignee:

SIRNA THERAPEUTICS, INC., Cambridge, MA (US);

Attorney:
Primary Examiner:
Int. Cl.
CPC ...
C07C 217/40 (2006.01); C12N 15/113 (2010.01); C07C 217/52 (2006.01); C07D 207/08 (2006.01); C07D 207/12 (2006.01); C07D 209/48 (2006.01); C07D 211/22 (2006.01); C07D 211/44 (2006.01); C07D 211/46 (2006.01); C07D 295/088 (2006.01); C07H 21/02 (2006.01);
U.S. Cl.
CPC ...
C12N 15/113 (2013.01); C07C 217/40 (2013.01); C07C 217/52 (2013.01); C07D 207/08 (2013.01); C07D 207/12 (2013.01); C07D 209/48 (2013.01); C07D 211/22 (2013.01); C07D 211/44 (2013.01); C07D 211/46 (2013.01); C07D 295/088 (2013.01); C07H 21/02 (2013.01); C12N 15/1137 (2013.01); C07C 2101/02 (2013.01); C12N 2310/14 (2013.01); C12N 2310/141 (2013.01); C12N 2310/321 (2013.01); C12N 2330/30 (2013.01);
Abstract

The instant invention provides for novel cationic lipids that can be used in combination with other lipid components such as cholesterol and PEG-lipids to form lipid nanoparticles with oligonucleotides. It is an object of the instant invention to provide a cationic lipid scaffold that is susceptible to hydrolytic instability that may translate into reduced liver residence times and reduced hepatocellular toxicity. The present invention employs acetals and ketals to provide a low pH sensitive chemical handle for degradation.


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