The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Nov. 01, 2016

Filed:

Apr. 04, 2012
Applicants:

Yoram Shechter, Rehovot, IL;

Matityahu Fridkin, Rehovot, IL;

Inventors:

Yoram Shechter, Rehovot, IL;

Matityahu Fridkin, Rehovot, IL;

Attorney:
Primary Examiner:
Int. Cl.
CPC ...
A61K 38/00 (2006.01); A61K 47/48 (2006.01); C07C 309/17 (2006.01); C07D 207/46 (2006.01); C07D 213/70 (2006.01); A61K 38/22 (2006.01); A61K 38/28 (2006.01); A61K 38/37 (2006.01); A61K 38/48 (2006.01);
U.S. Cl.
CPC ...
A61K 47/48038 (2013.01); A61K 38/22 (2013.01); A61K 38/28 (2013.01); A61K 38/37 (2013.01); A61K 38/4846 (2013.01); C07C 309/17 (2013.01); C07D 207/46 (2013.01); C07D 213/70 (2013.01); C12Y 304/21021 (2013.01);
Abstract

The present invention provides a long chain fatty acid (LCFA)-like albumin-binding probe/ligand containing no hydrolysable bond and having an enhanced associating affinity with human serum albumin, which upon conjugation with an amino- or mercapto-containing short-lived drug and administration of the conjugate, significantly prolongs the life time of said drug without substantially interfering with its pharmacological activity. The invention further provides conjugates of said probe with amino- or mercapto-containing drugs, as well as pharmaceutical compositions and uses thereof.


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