The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Oct. 18, 2016

Filed:

Jun. 15, 2015
Applicant:

The Trustees of Princeton University, Princeton, NJ (US);

Inventors:

Bonnie L. Bassler, Princeton, NJ (US);

Lee R. Swem, Montara, CA (US);

Scott M. Ulrich, Ithaca, NY (US);

Colleen T. O'Loughlin, San Francisco, CA (US);

Assignee:
Attorney:
Primary Examiner:
Assistant Examiner:
Int. Cl.
CPC ...
A01N 43/06 (2006.01); A61K 31/38 (2006.01); C07D 333/36 (2006.01); C07D 333/42 (2006.01); A61K 31/365 (2006.01); A01N 43/08 (2006.01); A01N 43/10 (2006.01); A01N 43/16 (2006.01); A01N 43/18 (2006.01); A61K 31/341 (2006.01); A61K 31/381 (2006.01); C07D 307/33 (2006.01);
U.S. Cl.
CPC ...
A61K 31/365 (2013.01); A01N 43/08 (2013.01); A01N 43/10 (2013.01); A01N 43/16 (2013.01); A01N 43/18 (2013.01); A61K 31/341 (2013.01); A61K 31/381 (2013.01); C07D 307/33 (2013.01); C07D 333/36 (2013.01);
Abstract

A novel small molecule antagonizes two types of acyl homoserine lactone receptors: membrane-bound and cytoplasmic. A focused library of analogs and derivatives of the original antagonist was synthesized. Analog and derivative molecules harbor a range of activities. The novel small molecule and most potent antagonist protects the eukaryotefrom quorum-sensing-mediated killing by the bacterial pathogen. The saving ofdemonstrates the use of these molecules as small molecule antimicrobials.


Find Patent Forward Citations

Loading…