The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Jan. 05, 2016

Filed:

Nov. 18, 2010
Applicants:

Anthony O. Chong, Huntsville, AL (US);

Seoju Lee, Madison, AL (US);

Bhalchandra V. Joshi, Madison, AL (US);

Brian Bray, Huntsville, AL (US);

Shaoyong Nie, Huntsville, AL (US);

Patrick L. Spence, Madison, AL (US);

Antoni Kozlowski, Huntsville, AL (US);

Samuel P. Mcmanus, Huntsville, AL (US);

Sachin Tipnis, Houston, TX (US);

David Swallow, Spring, TX (US);

John R. Handley, Duluth, MN (US);

Anthony G. Schaefer, Huntsville, AL (US);

Inventors:

Anthony O. Chong, Huntsville, AL (US);

Seoju Lee, Madison, AL (US);

Bhalchandra V. Joshi, Madison, AL (US);

Brian Bray, Huntsville, AL (US);

Shaoyong Nie, Huntsville, AL (US);

Patrick L. Spence, Madison, AL (US);

Antoni Kozlowski, Huntsville, AL (US);

Samuel P. McManus, Huntsville, AL (US);

Sachin Tipnis, Houston, TX (US);

Greg Lavaty, Sugar Land, TX (US);

David Swallow, Spring, TX (US);

John R. Handley, Duluth, MN (US);

Anthony G. Schaefer, Huntsville, AL (US);

Assignee:

Nektar Therapeutics, San Francisco, CA (US);

Attorneys:
Primary Examiner:
Int. Cl.
CPC ...
A61K 31/4745 (2006.01); C07D 491/22 (2006.01); A61K 47/48 (2006.01); C08G 65/329 (2006.01); C08G 65/333 (2006.01); C07C 51/41 (2006.01); C07C 53/18 (2006.01); C08G 65/48 (2006.01);
U.S. Cl.
CPC ...
A61K 47/48215 (2013.01); A61K 31/4745 (2013.01); C07C 51/412 (2013.01); C07C 53/18 (2013.01); C07D 491/22 (2013.01); C08G 65/329 (2013.01); C08G 65/33396 (2013.01); C08G 65/48 (2013.01); C08L 2203/02 (2013.01);
Abstract

Among other aspects, provided herein is a hydrohalide salt of a multi-arm water-soluble polyethylene glycol-drug conjugate, along with related methods of making and using the same. The hydrohalide salt is stably formed, and appears to be more resistant to hydrolytic degradation than the corresponding free base form of the conjugate.


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