The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Jul. 28, 2015

Filed:

Nov. 03, 2011
Applicants:

Ravi V. J. Chari, Newton, MA (US);

Wayne C. Widdison, Belmont, MA (US);

Sharon D. Wilhelm, Arlington, MA (US);

Inventors:

Ravi V. J. Chari, Newton, MA (US);

Wayne C. Widdison, Belmont, MA (US);

Sharon D. Wilhelm, Arlington, MA (US);

Assignee:

ImmunoGen, Inc., Waltham, MA (US);

Attorneys:
Primary Examiner:
Int. Cl.
CPC ...
A61K 39/00 (2006.01); C07D 498/16 (2006.01); A61K 47/48 (2006.01); A61K 45/06 (2006.01);
U.S. Cl.
CPC ...
C07D 498/16 (2013.01); A61K 45/06 (2013.01); A61K 47/48215 (2013.01); A61K 47/48384 (2013.01); A61K 47/48561 (2013.01);
Abstract

New ansamitocin derivatives bearing a linking group are disclosed. Also disclosed are methods for the synthesis of these new ansamitocin derivatives and methods for their linkage to cell-binding agents. The ansamitocin derivative-cell-binding agent conjugates are useful as therapeutic agents, which are delivered specifically to target cells and are cytotoxic. These conjugates display vastly improved therapeutic efficacy in animal tumor models compared to the previously described agents.


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