The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Patent No.:

US 7605259 B1

PDF
Full Text
Expired
Date of Patent:
Oct. 20, 2009

Filed:

Sep. 15, 2003
Applicants:

Amy Newman, Phoenix, MD (US);

Peter Grundt, Baltimore, MD (US);

Robert R. Luedtke, Fort Worth, TX (US);

Inventors:

Amy Newman, Phoenix, MD (US);

Peter Grundt, Baltimore, MD (US);

Robert R. Luedtke, Fort Worth, TX (US);

Attorney:
Primary Examiner:
Assistant Examiner:
Int. Cl.
CPC ...
C07D 241/04 (2006.01); C07D 295/00 (2006.01);
U.S. Cl.
CPC ...
Abstract

A family of structurally rigid dopamine D3 receptor selective ligands is described. The family of structurally rigid dopamine D3 receptor selective ligands has the formula wherein A is cis or trans —CH═CH—, —C═C—, or cyclohexyl. B is cis or trans —CH═CH— or absent. R1 represents an optionally substituted phenyl group, wherein said substituents are selected from the group consisting of: hydrogen, halogen, amino, nitro, hydroxyl, alkoxy, alkyl, acyl and pyridyl, and said substitution may occur at any of the ortho, meta, or para positions, or R1 represents a heteroaromatic ring. A preferred heteroaromatic ring is indole, quinoxoline, pyridyl, pyrimidyl, or imidazole. R2 and R3 may be independently hydrogen or a halogen, or R2 alone may be C1, C2, or C3 alkoxy, and m is 1 or 2, and n is 0, 1, or 2.


Find Patent Forward Citations

Newman, Amy. (2009). Structurally rigid dopamine d3 receptor selective ligands and process for making them (U.S. Patent No. 7605259). U.S. Patent and Trademark Office. https://idiyas.com/patent/badge/7605259

Data source: USPTO (United States Patent and Trademark Office) public patent records. Weekly synchronization. How IDiyas builds this profile

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