The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Nov. 18, 2025

Filed:

Mar. 24, 2020
Applicants:

Shanghai Synergy Pharmaceutical Sciences Co., Ltd., Shanghai, CN;

Zhejiang Huahai Pharmaceutical Co., Ltd., Zhejiang, CN;

Inventors:

Xin Xu, Shanghai, CN;

Jia Chen, Shanghai, CN;

Zhen Zhang, Shanghai, CN;

Liming Zhang, Shanghai, CN;

Qimei Wu, Shanghai, CN;

Qingyun Jiang, Shanghai, CN;

Fengying Guo, Shanghai, CN;

Yuyun Zhang, Shanghai, CN;

Hao Yu, Shanghai, CN;

Xiaojuan Zhang, Shanghai, CN;

Kang Sun, Shanghai, CN;

Xiaobo Zhou, Shanghai, CN;

Chengxu Zang, Shanghai, CN;

Yijin Wang, Shanghai, CN;

Xiaoer Xia, Shanghai, CN;

Yunfei Li, Shanghai, CN;

Jian Ge, Shanghai, CN;

Attorney:
Primary Examiner:
Assistant Examiner:
Int. Cl.
CPC ...
C07D 491/107 (2006.01); A61P 35/00 (2006.01); C07D 405/12 (2006.01); C07D 405/14 (2006.01); C07D 471/10 (2006.01); C07D 487/04 (2006.01); C07D 495/10 (2006.01);
U.S. Cl.
CPC ...
C07D 491/107 (2013.01); A61P 35/00 (2018.01); C07D 405/12 (2013.01); C07D 405/14 (2013.01); C07D 471/10 (2013.01); C07D 487/04 (2013.01); C07D 495/10 (2013.01);
Abstract

Provided are amide compounds, a preparation method therefor, and use thereof in the medical field. Specifically, provided are small molecule amide compounds. Such compounds are inhibitors of enhancer of Zeste homolog 2 (EZH2), and can be used for preventing and/or treating related diseases mediated by EZH2, including tumors, myeloproliferative diseases or autoimmune diseases.


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