The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Dec. 05, 2023

Filed:

Oct. 02, 2020
Applicant:

Nektar Therapeutics, San Francisco, CA (US);

Inventors:

Antoni Kozlowski, Huntsville, AL (US);

Samuel P. McManus, Huntsville, AL (US);

Sachin Tipnis, Houston, TX (US);

Greg Lavaty, Sugar Land, TX (US);

David Swallow, Spring, TX (US);

John R. Handley, Eveleth, MN (US);

Anthony G. Schaefer, Huntsville, AL (US);

Assignee:

Nektar Therapeutics, San Francisco, CA (US);

Attorney:
Primary Examiner:
Assistant Examiner:
Int. Cl.
CPC ...
C08G 65/331 (2006.01); C08G 65/329 (2006.01); C08G 65/333 (2006.01); A61K 47/60 (2017.01); C08G 65/48 (2006.01); C07D 491/22 (2006.01); C07C 51/41 (2006.01); C07C 53/18 (2006.01); A61K 31/4745 (2006.01);
U.S. Cl.
CPC ...
C08G 65/331 (2013.01); A61K 31/4745 (2013.01); A61K 47/60 (2017.08); C07C 51/412 (2013.01); C07C 53/18 (2013.01); C07D 491/22 (2013.01); C08G 65/329 (2013.01); C08G 65/33396 (2013.01); C08G 65/48 (2013.01); C08L 2203/02 (2013.01);
Abstract

Among other aspects, provided herein is a mixed-acid salt of a water-soluble polymer-drug conjugate, along with related methods of making and using the same. The mixed-salt acid salt is stably formed, and appears to be more resistant to hydrolytic degradation than the corresponding predominantly pure acid salt or free base forms of the polymer-drug conjugate. The mixed acid salt is reproducibly prepared and recovered, and provides surprising advantages over non-mixed acid salt forms of the water-soluble polymer drug conjugate.


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