The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Nov. 05, 2019

Filed:

Mar. 03, 2017
Applicant:

Bionevia Pharmaceuticals, Inc., Cambridge, MA (US);

Inventors:

Isabel Kalofonos, Cambridge, MA (US);

G. Patrick Stahly, West Lafayette, IN (US);

William Martin-Doyle, Cambridge, MA (US);

Dimitris Kalofonos, Cambridge, MA (US);

Travis L. Houston, Lafayette, IN (US);

Jeffrey S. Stults, West Lafayette, IN (US);

Assignee:

BIONEVIA PHARMACEUTICALS, INC., Cambridge, MA (US);

Attorney:
Primary Examiner:
Int. Cl.
CPC ...
A61K 31/427 (2006.01); C07D 277/36 (2006.01); A61K 31/14 (2006.01); A61K 31/426 (2006.01); C07C 215/40 (2006.01);
U.S. Cl.
CPC ...
C07D 277/36 (2013.01); A61K 31/14 (2013.01); A61K 31/426 (2013.01); A61K 31/427 (2013.01); C07C 215/40 (2013.01); C07B 2200/13 (2013.01);
Abstract

The invention relates to a novel choline cocrystal of 5-[(1Z.2E)-2-methyl-3-phenylpropenylidene]-4-oxo-2-thioxo-3-thiazolidineacetic acid. The preparation and characterization of the novel choline cocrystal according to various embodiments of the invention is described. The invention also relates to pharmaceutical compositions containing the novel choline cocrystal and the therapeutic use of the novel choline cocrystal to treat and/or prevent various conditions, including treating and/or preventing diabetic complications, treating and/or preventing homocystinuria reducing levels of homocysteine in blood serum, inhibiting aldose reductase, and affording cardioprotection in non-diabetic patients.


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