The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Jul. 31, 2018

Filed:

Jun. 15, 2017
Applicant:

Eli Lilly and Company, Indianapolis, IN (US);

Inventors:

Michael Edward Kobierski, Greenwood, IN (US);

Michael E. Kopach, Greenwood, IN (US);

Pingyun Chen, Chapel Hill, NC (US);

Assignee:

ELI LILLY AND COMPANY, Indianapolis, IN (US);

Attorney:
Primary Examiner:
Int. Cl.
CPC ...
C07D 401/14 (2006.01); C07D 401/06 (2006.01); C07D 213/53 (2006.01); C07D 213/50 (2006.01);
U.S. Cl.
CPC ...
C07D 401/06 (2013.01); C07D 213/50 (2013.01); C07D 213/53 (2013.01); C07D 401/14 (2013.01);
Abstract

The present invention relates to novel compounds, (2-chlorophenyl)-[2-(2-hydroxy-2-pyridin-4-yl-vinyl)pyridin-3-yl]methanone benzoate, and (2-chlorophenyl)-[2-(2-hydroxy-2-pyridin-4-yl-vinyl)pyridin-3-yl]methanone toluate, which are useful intermediates for the preparation of the compound of Formula I: The present invention further relates to novel processes for preparing a crystalline compound, which is {2-[1-(3,5-bis-trifluoromethyl-benzyl)-5-pyridin-4-yl-1H-[1,2,3]triazol-4-yl]-pyridin-3-yl}-(2-chlorophenyl)-methanone, Form IV.


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