The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Jun. 05, 2018

Filed:

Mar. 18, 2015
Applicant:

Mayo Foundation for Medical Education and Research, Rochester, MN (US);

Inventors:

Timothy R. Degrado, Rochester, MN (US);

Huailel Jiang, Rochester, MN (US);

Attorney:
Primary Examiner:
Int. Cl.
CPC ...
C07C 51/60 (2006.01); A61K 51/04 (2006.01);
U.S. Cl.
CPC ...
C07C 51/60 (2013.01); A61K 51/0402 (2013.01);
Abstract

Methods, compositions, and systems related to preparing gaseousF-compounds for use in radiolabeling positron emission tomography (PET) tracer precursor compounds are disclosed. [F]fluoride ions produced by conventional methods are converted by reaction with an acid anhydride having the formula: to a gaseousF-compound having the formula: wherein each R is independently a substituted or unsubstituted, straight chain or branched C-Calkyl group. The gaseousF-compounds, which also can be readily trapped on solid-phase extraction media or in organic solvents such as acetonitrile, provide an alternative source of [F]fluoride for use in the nucleophilic substitution reactions that are used to synthesize a large number ofF-labeled PET imaging tracers, including 2-[F]fluoro-2-deoxyglucose (FDG).


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