The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Apr. 10, 2018

Filed:

Nov. 19, 2014
Applicant:

Hiroshi Maeda, Kumamcto, JP;

Inventors:

Hiroshi Maeda, Kumamoto, JP;

Hideaki Nakamura, Kumamoto, JP;

Jun Fang, Kumamoto, JP;

Assignee:

Other;

Attorney:
Primary Examiner:
Assistant Examiner:
Int. Cl.
CPC ...
C08F 222/06 (2006.01); C08F 8/44 (2006.01); C08F 8/42 (2006.01); C08F 8/34 (2006.01); C08F 8/12 (2006.01); C08F 8/32 (2006.01); C08F 8/30 (2006.01); A61K 38/00 (2006.01); C07K 14/575 (2006.01); A61K 31/409 (2006.01); A61K 31/69 (2006.01); A61K 31/704 (2006.01); C08F 220/04 (2006.01); A61K 47/58 (2017.01);
U.S. Cl.
CPC ...
A61K 31/409 (2013.01); A61K 31/69 (2013.01); A61K 31/704 (2013.01); A61K 47/58 (2017.08); C08F 8/12 (2013.01); C08F 8/30 (2013.01); C08F 8/32 (2013.01); C08F 8/34 (2013.01); C08F 8/42 (2013.01); C08F 8/44 (2013.01); C08F 220/04 (2013.01); C08F 222/06 (2013.01); A61K 38/00 (2013.01); C07K 14/575 (2013.01); C08F 2800/10 (2013.01);
Abstract

The present invention provides a group of novel SMA derivatives and a covalent conjugate of the derivatives and an active substance. More specifically, the present invention provides: an SMA derivative which contains (i) a styrene-maleic acid copolymer (SMA) and (ii) a side chain (b) that contains a functional group (a) selected from among —NH2, —SH, —OH, —COOH, —NH—(C═NH)—NHand —C(CH—OH)and introduced into a carboxyl group of a maleic acid residue of the SMA via an amide bond or an ester bond, and wherein when a plurality of side chain (b) is introduced into the SMA, the side chains (b) may be identical or different from each other; and a conjugate of this SMA derivative and an active substance.


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