The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.
The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.
Patent No.:
Date of Patent:
Mar. 27, 2018
Filed:
May. 29, 2015
Applicant:
Tetrahedron, Paris, FR;
Inventors:
Irene Erdelmeier, Paris, FR;
Sylvain Daunay, Paris, FR;
Assignee:
TETRAHEDRON, Paris, FR;
Attorney:
Primary Examiner:
Int. Cl.
CPC ...
C07D 233/84 (2006.01); C07D 403/12 (2006.01);
U.S. Cl.
CPC ...
C07D 403/12 (2013.01); C07D 233/84 (2013.01);
Abstract
The invention relates to a compound of the 5-acylsulfanyl-histidine type and the derivatives thereof, of general formula (I), wherein R1 to R3=H, alkyl, especially CH3; R4=H, alkyl, especially CH3, alkyle(C=0), substituted alkyl (C═O), aryl (C═O); β-alanyl (H2NCH2CH2 (C═O); α-amino-acyl; R5=alkyl, especially methyl, phenyl. The invention also relates to the use of said compound for producing compounds of the 5-sulfanyl-histidine type and the derivatives thereof, in addition to corresponding disulfides; and to the various methods for the production thereof.