The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Mar. 20, 2018

Filed:

Aug. 26, 2016
Applicants:

Novartis Ag, Basel, CH;

Massachusetts Institute of Technology, Cambridge, MA (US);

Inventors:

Naresh Chennamsetty, Cambridge, MA (US);

Bernhard Helk, Basel, CH;

Bernhardt Trout, Cambridge, MA (US);

Veysel Kayser, Cambridge, MA (US);

Vladimir Voynov, Cambridge, MA (US);

Assignees:

Novartis AG, Basel, CH;

Massachusetts Institute of Technology, Cambridge, MA (US);

Attorney:
Primary Examiner:
Int. Cl.
CPC ...
G06F 19/16 (2011.01); C07K 14/71 (2006.01); C07K 16/00 (2006.01); G06F 19/24 (2011.01); G06F 19/00 (2018.01); A61K 38/00 (2006.01);
U.S. Cl.
CPC ...
G06F 19/16 (2013.01); C07K 14/71 (2013.01); C07K 16/00 (2013.01); A61K 38/00 (2013.01); C07K 2317/94 (2013.01); G06F 19/24 (2013.01); G06F 19/70 (2013.01);
Abstract

The present invention provides methods and computational tools based, at least in part, on computer simulations that identify macromolecule binding regions and aggregation prone regions of a protein. Substitutions may then be made in these aggregation prone regions to engineer proteins with enhanced stability and/or a reduced propensity for aggregation. Similarly, substitutions may then be made in these macromolecule binding regions to engineer proteins with altered binding affinity for the macromolecule.


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