The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Jan. 30, 2018

Filed:

May. 13, 2015
Applicant:

Memorial Sloan Kettering Cancer Center, New York, NY (US);

Inventors:

Gabriela Chiosis, New York, NY (US);

Yanlong Kang, Plainsboro, NJ (US);

Hardik J. Patel, Kew Gardens, NY (US);

Maulik Patel, New York, NY (US);

Stefan Ochiana, Chevy Chase, MD (US);

Anna Rodina, New York, NY (US);

Tony Taldone, Forest Hills, NY (US);

Liza Shrestha, New York, NY (US);

Assignee:
Attorneys:
Primary Examiner:
Int. Cl.
CPC ...
C07D 239/46 (2006.01); A61K 31/506 (2006.01); C07D 405/12 (2006.01); C07D 401/12 (2006.01); C07D 403/04 (2006.01); C07D 417/12 (2006.01); C07D 413/12 (2006.01); C07D 407/12 (2006.01); A61K 31/5377 (2006.01); A61K 45/06 (2006.01);
U.S. Cl.
CPC ...
C07D 239/46 (2013.01); A61K 31/506 (2013.01); A61K 31/5377 (2013.01); A61K 45/06 (2013.01); C07D 401/12 (2013.01); C07D 403/04 (2013.01); C07D 405/12 (2013.01); C07D 407/12 (2013.01); C07D 413/12 (2013.01); C07D 417/12 (2013.01);
Abstract

The present invention provides compounds I and II and compositions thereof for use in the modulation of Hsp70. In some embodiments, the present invention provides a method for inhibiting Hsp70 activity. In some embodiments, the present invention provides a method of treating a subject suffering from or susceptible to a disease, disorder, or condition responsive to Hsp70 inhibition comprising administering to the subject a therapeutically effective amount of a provided compound. In some embodiments, the present invention provides a method for treating or preventing cancer in a subject suffering therefrom, comprising administering to a patient in need thereof a therapeutically effective amount of a provided compound.


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