The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Dec. 26, 2017

Filed:

Jun. 22, 2015
Applicant:

Reiley Pharmaceuticals, Inc., San Jose, CA (US);

Inventors:

Mark A. Reiley, Washington, DC (US);

B. Michael Silber, San Francisco, CA (US);

Julio Medina, San Carlos, CA (US);

Frank Kayser, San Francisco, CA (US);

William D. Shrader, Belmont, CA (US);

Assignee:

Reiley Pharmaceuticals, Inc., San Jose, CA (US);

Attorney:
Primary Examiner:
Assistant Examiner:
Int. Cl.
CPC ...
A61M 36/00 (2006.01); A61K 51/00 (2006.01); C07B 59/00 (2006.01); C07F 13/00 (2006.01); A61K 51/04 (2006.01);
U.S. Cl.
CPC ...
C07B 59/004 (2013.01); A61K 51/0402 (2013.01); A61K 51/0478 (2013.01); A61K 51/0487 (2013.01); A61K 51/0497 (2013.01); C07F 13/00 (2013.01); C07F 13/005 (2013.01);
Abstract

Conjugates derived from non-steroidal anti-inflammatory drugs (NSAIDs) and methods of use thereof are disclosed, useful for, inter alia, identifying and localizing the site of pathology and/or inflammation responsible for the sensation of pain in a patient; for identifying the sites of primary, secondary, benign, or malignant tumors; and for diagnosing infection or confirming or ruling out suspected infection. The NSAID-based conjugates contain an imaging moiety. The conjugates concentrate at sites of increased cyclooxygenase expression, thus revealing the sites of increased prostaglandin production, which is correlated with pain and inflammation, and correlated with tumor presence and/or location. Identifying areas of increased COX expressing can also aid in screening for infections.


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