The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Nov. 07, 2017

Filed:

Jan. 26, 2016
Applicant:

Fundación Centro Nacional DE Investigaciones Oncologicas Carlos Iii, Madrid, ES;

Attorneys:
Primary Examiner:
Int. Cl.
CPC ...
A61K 45/06 (2006.01); A61K 31/5383 (2006.01); C07D 513/16 (2006.01); C07D 513/22 (2006.01); C07D 515/22 (2006.01); A61K 31/4375 (2006.01); A61K 31/439 (2006.01); A61K 31/4745 (2006.01); A61K 31/5025 (2006.01); A61K 31/519 (2006.01);
U.S. Cl.
CPC ...
A61K 31/5383 (2013.01); A61K 31/439 (2013.01); A61K 31/4375 (2013.01); A61K 31/4745 (2013.01); A61K 31/5025 (2013.01); A61K 31/519 (2013.01); A61K 45/06 (2013.01); C07D 513/16 (2013.01); C07D 513/22 (2013.01); C07D 515/22 (2013.01);
Abstract

There is provided compounds of formula I, wherein R1, R, R, R, X, Y, Z, Rand ring A/B have meanings given in the description, and pharmaceutically-acceptable esters, amides, solvates or salts thereof, which compounds are useful in the treatment of diseases in which inhibition of a protein or lipid kinase (e.g. PI3-K, particularly class I PI3K, PIM family kinase and/or mTOR) is desired and/or required, and particularly in the treatment of cancer. The invention also relates to combinations containing such compounds.


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