The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Aug. 29, 2017

Filed:

Feb. 26, 2016
Applicant:

Salk Institute for Biological Studies, La Jolla, CA (US);

Inventors:

David R. Schubert, La Jolla, CA (US);

Pamela A. Maher, La Jolla, CA (US);

Chandramouli Chiruta, La Jolla, CA (US);

Assignee:
Attorney:
Primary Examiner:
Assistant Examiner:
Int. Cl.
CPC ...
A61K 31/4025 (2006.01); C07D 311/78 (2006.01); A61K 31/47 (2006.01); C07D 311/30 (2006.01); A61K 31/4709 (2006.01); A61K 31/452 (2006.01); C07D 311/62 (2006.01); C07D 215/233 (2006.01); A61K 45/06 (2006.01); A61K 31/12 (2006.01); A61K 31/352 (2006.01); A61K 31/353 (2006.01); C07C 49/835 (2006.01); C07C 49/84 (2006.01); C07D 311/60 (2006.01);
U.S. Cl.
CPC ...
A61K 31/47 (2013.01); A61K 31/12 (2013.01); A61K 31/352 (2013.01); A61K 31/353 (2013.01); A61K 31/4025 (2013.01); A61K 31/4709 (2013.01); A61K 45/06 (2013.01); C07C 49/835 (2013.01); C07C 49/84 (2013.01); C07D 215/233 (2013.01); C07D 311/30 (2013.01); C07D 311/60 (2013.01); C07D 311/62 (2013.01); C07D 311/78 (2013.01);
Abstract

The present invention provides neuroprotective polyphenol compounds, which can be synthetic analogs of fisetin, baicalein or chlorogenic acid, that maintain neuroprotective, anti-inflammatory, glutathione promoting, and/or antioxidant properties. The neuroprotective polyphenol compounds are useful for promoting, enhancing and/or increasing neuron protection, growth and/or regeneration. The polyphenol compounds further find use for increasing and or maintaining intracellular glutathione (GSH) levels. The polyphenol compounds are also useful for treating, preventing, mitigating and/or delaying neurodegenerative conditions, including diabetes, Parkinson's disease, Huntington's disease, Alzheimer's disease, non-Alzheimer's dementias, multiple sclerosis, traumatic brain injury, spinal cord injury or ALS.


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