The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
May. 23, 2017

Filed:

Oct. 09, 2013
Applicant:

Aston University, Birmingham, GB;

Inventors:

Martin Griffin, Bleasby, GB;

Daniel Rathbone, Conventry, GB;

Leonas Eduard Badarau, Villenave D'Ornon, FR;

Assignee:

ASTON UNIVERSITY, Birmingham, GB;

Attorneys:
Primary Examiner:
Assistant Examiner:
Int. Cl.
CPC ...
A61K 31/495 (2006.01); A61P 25/28 (2006.01); A61P 31/18 (2006.01); A61P 17/06 (2006.01); A61P 7/02 (2006.01); A61P 29/00 (2006.01); C07D 295/26 (2006.01); C07D 233/84 (2006.01); C07D 295/185 (2006.01); C07D 295/205 (2006.01);
U.S. Cl.
CPC ...
C07D 295/26 (2013.01); C07D 233/84 (2013.01); C07D 295/185 (2013.01); C07D 295/205 (2013.01);
Abstract

The present invention relates to novel compounds of Formula I capable of inhibiting tissue transglutaminase, and uses of the same in medicine. In particular, the invention provides compounds for use in the treatment of prevention of disease and conditions such as fibrosis (e.g. cystic fibrosis), scarring, neurodegenerative diseases (e.g. Alzheimer's disease, Huntington's disease and Parkinson's disease), autoimmune diseases (e.g. multiple sclerosis and coeliac disease), thrombosis, proliferative disorders (e.g. cancers), AIDS, psoriasis and inflammation (e.g. chronic inflammatory diseases).


Find Patent Forward Citations

Loading…