The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.
The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.
Patent No.:
Date of Patent:
May. 16, 2017
Filed:
Jan. 11, 2013
Applicant:
Medeia Therapeutics Ltd, Kuopio, FI;
Inventors:
Assignee:
ARANDA PHARMA LTD, Kuopio, FI;
Attorney:
Primary Examiner:
Assistant Examiner:
Int. Cl.
CPC ...
A01N 43/58 (2006.01); A61K 31/60 (2006.01); A61K 31/50 (2006.01); A61K 31/495 (2006.01); A01N 43/40 (2006.01); A61K 31/44 (2006.01); C07D 487/00 (2006.01); C07D 213/00 (2006.01); C07D 211/78 (2006.01); C07D 211/90 (2006.01); C07D 213/84 (2006.01); C07D 487/04 (2006.01); C07D 213/30 (2006.01); C07D 213/57 (2006.01); C07D 213/61 (2006.01); A61K 31/435 (2006.01); A61K 31/444 (2006.01); A61K 31/5025 (2006.01); C07D 213/89 (2006.01); C07D 401/06 (2006.01);
U.S. Cl.
CPC ...
C07D 487/04 (2013.01); A61K 31/435 (2013.01); A61K 31/444 (2013.01); A61K 31/5025 (2013.01); C07D 213/30 (2013.01); C07D 213/57 (2013.01); C07D 213/61 (2013.01); C07D 213/89 (2013.01); C07D 401/06 (2013.01);
Abstract
The invention relates to novel heteroarylamide derivatives having formula (I) and N-oxides, stereoisomers and pharmaceutically acceptable salts thereof, where R, R, R1 1, R', R″, z and X are as defined in the claims. The arylamide derivatives of formula (I) have antiandrogenic properties. The invention also relates to compounds of formula (I) for use as a medicament and to pharmaceutical compositions comprising them and to their preparation.