The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
May. 09, 2017

Filed:

Apr. 22, 2014
Applicant:

The General Hospital Corporation, Boston, MA (US);

Inventors:

Robert Zahler, Pennington, NJ (US);

Ronald Thure Wester, Ledyard, CT (US);

Steven Joseph Brickner, Ledyard, CT (US);

Attorney:
Primary Examiner:
Assistant Examiner:
Int. Cl.
CPC ...
C07D 235/08 (2006.01); C07D 235/28 (2006.01); C07D 401/12 (2006.01); C07D 403/12 (2006.01); C07D 235/16 (2006.01); C07D 235/26 (2006.01); C07D 235/30 (2006.01); C07D 403/04 (2006.01); C07D 405/12 (2006.01); C07D 413/04 (2006.01); C07D 413/12 (2006.01); C07D 471/04 (2006.01); C07D 263/58 (2006.01); C07D 417/12 (2006.01);
U.S. Cl.
CPC ...
C07D 235/28 (2013.01); C07D 235/16 (2013.01); C07D 235/26 (2013.01); C07D 235/30 (2013.01); C07D 263/58 (2013.01); C07D 401/12 (2013.01); C07D 403/04 (2013.01); C07D 403/12 (2013.01); C07D 405/12 (2013.01); C07D 413/04 (2013.01); C07D 413/12 (2013.01); C07D 417/12 (2013.01); C07D 471/04 (2013.01);
Abstract

The disclosure provides compounds and pharmaceutical compositions of the compounds useful for treating chronic and acute bacterial infections. Certain of the compounds are compounds and salts of general Formula VIII Certain compounds of this disclosure are MvfR inhibitors. MvfR inhibitors reduce the formation of antibiotic tolerant bacterial strains and are useful for treating Gram-negative bacterial infections and reducing the virulence of. Methods of treating bacterial infections in a patient, includinginfections, are also provided by the disclosure.


Find Patent Forward Citations

Loading…