The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Mar. 28, 2017

Filed:

Jul. 29, 2013
Applicant:

Riken, Wako-shi, Saitama, JP;

Inventors:

Fumihiko Ishikawa, Saitama, JP;

Yoriko Saito, Wako, JP;

Yoshinobu Hashizume, Wako, JP;

Yasuko Koda, Wako, JP;

Hitomi Yuki, Wako, JP;

Assignee:

RIKEN, Saitama, JP;

Attorney:
Int. Cl.
CPC ...
C07D 487/04 (2006.01); A61K 31/519 (2006.01); A61K 31/4985 (2006.01); A61P 35/02 (2006.01); A61K 45/06 (2006.01); A61K 31/4709 (2006.01); A61K 31/7105 (2006.01); A61K 31/713 (2006.01); C07D 519/00 (2006.01); C12Q 1/68 (2006.01);
U.S. Cl.
CPC ...
C07D 487/04 (2013.01); A61K 31/4709 (2013.01); A61K 31/4985 (2013.01); A61K 31/519 (2013.01); A61K 31/713 (2013.01); A61K 31/7105 (2013.01); A61K 45/06 (2013.01); C07D 519/00 (2013.01); C12Q 1/6886 (2013.01); C12Q 2600/106 (2013.01); C12Q 2600/156 (2013.01); C12Q 2600/16 (2013.01);
Abstract

This invention relates to an agent for treating or inhibiting recurrence of acute myeloid leukemia and an agent for inhibiting growth of leukemia stem cells comprising a compound represented by formula (I) or a salt thereof: wherein Arand Areach represent aryl or heteroaryl; L represents O, S, NH, NHCO, or CONH; X represents CH or N; Y represents C-alkylene; Zrepresents hydrogen, C-alkyl, amino-C-alkyl, C-alkylamino-C-alkyl, di(C-alkyl)amino-C-alkyl, hydroxy-C-alkyl, C-alkoxy-C-alkyl, or carboxy-C-alkyl; and Zrepresents C-alkyl, amino-C-alkyl, C-alkylamino-C-alkyl, di(C-alkyl)amino-C-alkyl, hydroxy-C-alkyl, C-alkoxy-C-alkyl, or carboxy-C-alkyl, Zand Zmay, together with adjacent nitrogen, form a heterocyclic group containing as a ring member one or more hetero atoms, in addition to the nitrogen adjacent to Zand Z.


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