The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.
The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.
Patent No.:
Date of Patent:
Mar. 07, 2017
Filed:
Aug. 26, 2013
Applicants:
Shanghai Hengrui Pharmaceutical Co., Ltd., Shanghai, CN;
Jiangsu Hengrui Medicine Co., Ltd., Lianyungang, Jiangsu, CN;
Inventors:
Hejun Lu, Shanghai, CN;
Piaoyang Sun, Lianyungang, CN;
Hongbo Fei, Shanghai, CN;
Hongjian Jiang, Shanghai, CN;
Haowei Wang, Shanghai, CN;
Qing Dong, Shanghai, CN;
Assignees:
Shanghai Hengrui Pharmaceutical Co., Ltd., Shanghai, CN;
Jiangsu Hengrui Medicine Co., Ltd., Lianyungang, Jiangsu, CN;
Primary Examiner:
Int. Cl.
CPC ...
C07D 233/86 (2006.01); C07D 409/12 (2006.01); C07D 403/12 (2006.01); C07D 405/14 (2006.01); C07D 405/12 (2006.01); C07D 401/04 (2006.01); C07D 401/12 (2006.01);
U.S. Cl.
CPC ...
C07D 409/12 (2013.01); C07D 233/86 (2013.01); C07D 401/04 (2013.01); C07D 401/12 (2013.01); C07D 403/12 (2013.01); C07D 405/12 (2013.01); C07D 405/14 (2013.01);
Abstract
New imidazoline derivatives represented by formula (I): preparation methods thereof, pharmaceutical compositions comprising such derivatives, and applications of such derivatives in preparing androgen receptor antagonists and medicaments for treating diseases such as prostate cancer are described.