The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Feb. 14, 2017

Filed:

Nov. 01, 2013
Applicants:

Whitehead Institute for Biomedical Research, Cambridge, MA (US);

Dana-farber Cancer Institute, Inc., Boston, MA (US);

Inventors:

James E. Bradner, Weston, MA (US);

Michael R. McKeown, Brookline, MA (US);

Peter B. Rahl, Natick, MA (US);

Richard A. Young, Boston, MA (US);

Jason J. Marineau, Franklin, MA (US);

Attorney:
Primary Examiner:
Int. Cl.
CPC ...
C07D 207/327 (2006.01); C07D 401/12 (2006.01); C07D 207/27 (2006.01); C07D 209/04 (2006.01); C07D 403/06 (2006.01); C07D 409/04 (2006.01); C07D 413/12 (2006.01); C07D 417/06 (2006.01);
U.S. Cl.
CPC ...
C07D 207/327 (2013.01); C07D 207/27 (2013.01); C07D 209/04 (2013.01); C07D 401/12 (2013.01); C07D 403/06 (2013.01); C07D 409/04 (2013.01); C07D 413/12 (2013.01); C07D 417/06 (2013.01);
Abstract

The present invention provides compounds of Formula (I-A), (I-B), and (I-C), pharmaceutically acceptable salts thereof, and pharmaceutical compositions thereof. Compounds of the present invention are useful for inhibiting Myc (e.g., c-Myc) activity. The present invention further provides methods of using the compounds described herein for treating Myc-mediated disorders (e.g., cancer and other proliferative diseases). The present invention also provides assays for identifying Myc inhibitors.


Find Patent Forward Citations

Loading…