The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Patent No.:

US 9556113 B1

PDF
Full Text
Expired
Date of Patent:
Jan. 31, 2017

Filed:

Apr. 29, 2015
Applicants:

The South Dakota Board of Regents, Pierre, SD (US);

Sanford Research, Sioux Falls, SD (US);

Inventors:

Xiangming Guan, Brookings, SD (US);

Chandrahar Dwivedi, Brookings, SD (US);

Yinghong Li, Beijing, CN;

Yang Yang, Brookings, SD (US);

John H. Lee, Sioux Falls, SD (US);

Wilson Keith Miskimins, Alcester, SD (US);

Assignees:

The South Dakota Board of Regents, Pierre, SD (US);

Sanford Research, Sioux Falls, SD (US);

Attorneys:
Primary Examiner:
Int. Cl.
CPC ...
C07C 235/74 (2006.01); A61K 45/06 (2006.01); A61N 5/10 (2006.01); A61K 31/225 (2006.01); C07C 233/56 (2006.01); A61K 33/24 (2006.01); A61K 9/00 (2006.01); A61K 47/02 (2006.01); A61K 47/10 (2006.01); A61K 47/14 (2006.01); A61K 47/18 (2006.01); A61K 47/26 (2006.01); A61K 9/06 (2006.01); A61K 47/32 (2006.01); A61K 9/08 (2006.01); A61K 47/38 (2006.01); A61K 47/44 (2006.01); A61K 9/20 (2006.01); A61K 9/48 (2006.01);
U.S. Cl.
CPC ...
C07C 235/74 (2013.01); A61K 9/008 (2013.01); A61K 9/0019 (2013.01); A61K 9/06 (2013.01); A61K 9/08 (2013.01); A61K 9/2018 (2013.01); A61K 9/2027 (2013.01); A61K 9/2054 (2013.01); A61K 9/2059 (2013.01); A61K 9/4858 (2013.01); A61K 9/4866 (2013.01); A61K 31/225 (2013.01); A61K 33/24 (2013.01); A61K 45/06 (2013.01); A61K 47/02 (2013.01); A61K 47/10 (2013.01); A61K 47/14 (2013.01); A61K 47/18 (2013.01); A61K 47/26 (2013.01); A61K 47/32 (2013.01); A61K 47/38 (2013.01); A61K 47/44 (2013.01); A61N 5/10 (2013.01); C07C 233/56 (2013.01); A61N 2005/1098 (2013.01);
Abstract

The invention novel compounds, pharmaceutical compositions and methods useful for preventing or treating cancer in animals and humans. Also, the invention provides novel prodrugs useful for reducing tumor size, and inhibiting the growth of cancers, inhibiting tumor cell growth and tumor cell proliferation, and promoting apoptosis of tumor cells. When used in combination with chemoradiation therapy, the novel compounds, compositions and prodrugs provided herein can improve the effectiveness of chemoradiation therapy. The novel compounds, compositions and prodrugs of the invention inhibit PDK and LDH in unique and effective ways.


Find Patent Forward Citations

Loading…