The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Dec. 20, 2016

Filed:

Mar. 14, 2014
Applicant:

Zymeworks Inc., Vancouver, CA;

Inventors:

Geoffrey C. Winters, Vancouver, CA;

Alexander L. Mandel, Vancouver, CA;

Bradley J. Hedberg, Vancouver, CA;

John Babcook, Vancouver, CA;

James R. Rich, Vancouver, CA;

Tom Han Hsiao Hsieh, Vancouver, CA;

Elyse Marie Josée Bourque, Blaine, WA (US);

Assignee:

ZYMEWORKS INC., Vancouver, BC, unknown;

Attorneys:
Primary Examiner:
Int. Cl.
CPC ...
C07C 311/51 (2006.01); C07C 323/67 (2006.01); C07C 381/08 (2006.01); C07C 327/06 (2006.01); C07C 323/12 (2006.01); C07D 207/452 (2006.01); C07D 211/34 (2006.01); C07D 207/08 (2006.01); C07D 333/34 (2006.01); C07D 213/56 (2006.01); C07D 211/60 (2006.01); C07D 213/71 (2006.01); C07K 5/027 (2006.01); C07K 5/065 (2006.01); A61K 38/05 (2006.01); A61K 38/06 (2006.01); A61K 31/445 (2006.01); A61K 39/395 (2006.01); A61K 47/48 (2006.01); C07K 5/02 (2006.01); C07C 317/28 (2006.01); C07C 317/32 (2006.01); C07C 317/50 (2006.01);
U.S. Cl.
CPC ...
C07C 311/51 (2013.01); A61K 31/445 (2013.01); A61K 38/05 (2013.01); A61K 38/06 (2013.01); A61K 39/3955 (2013.01); A61K 47/48261 (2013.01); A61K 47/48415 (2013.01); C07C 323/12 (2013.01); C07C 323/67 (2013.01); C07C 327/06 (2013.01); C07C 381/08 (2013.01); C07D 207/08 (2013.01); C07D 207/452 (2013.01); C07D 211/34 (2013.01); C07D 211/60 (2013.01); C07D 213/56 (2013.01); C07D 213/71 (2013.01); C07D 333/34 (2013.01); C07K 5/0205 (2013.01); C07K 5/06078 (2013.01); C07C 317/28 (2013.01); C07C 317/32 (2013.01); C07C 317/50 (2013.01); C07C 2101/02 (2013.01); C07C 2101/08 (2013.01); C07C 2101/14 (2013.01);
Abstract

Compounds having cytotoxic and/or anti-mitotic activity are disclosed. The compounds have the following structure (I): including stereoisomers, pharmaceutically acceptable salts and prodrugs thereof, wherein R, R, R, Rand Rare as defined herein. Methods associated with preparation and use of such compounds, as well as pharmaceutical compositions comprising such compounds, are also disclosed. Also disclosed are compositions having the structure: (T)-(L)-(D), wherein (T) is a targeting moiety, (L) is an optional linker, and (D) is a compound having structure (I).


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