The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Nov. 01, 2016

Filed:

Sep. 10, 2010
Applicants:

Christopher J Creighton, San Diego, CA (US);

Leslie William Tari, San Diego, CA (US);

Zhiyong Chen, San Diego, CA (US);

Mark Hilgers, San Diego, CA (US);

Thanh to Lam, San Diego, CA (US);

Xiaoming LI, San Diego, CA (US);

Michael Trzoss, San Diego, CA (US);

Junhu Zhang, San Diego, CA (US);

John Finn, San Diego, CA (US);

Daniel Bensen, Carlsbad, CA (US);

Inventors:

Christopher J Creighton, San Diego, CA (US);

Leslie William Tari, San Diego, CA (US);

Zhiyong Chen, San Diego, CA (US);

Mark Hilgers, San Diego, CA (US);

Thanh To Lam, San Diego, CA (US);

Xiaoming Li, San Diego, CA (US);

Michael Trzoss, San Diego, CA (US);

Junhu Zhang, San Diego, CA (US);

John Finn, San Diego, CA (US);

Daniel Bensen, Carlsbad, CA (US);

Assignee:

Merck Sharp & Dohme Corp., Rahway, NJ (US);

Attorneys:
Primary Examiner:
Assistant Examiner:
Int. Cl.
CPC ...
C07D 487/04 (2006.01); C07D 519/00 (2006.01); C07D 471/04 (2006.01); C07D 487/16 (2006.01); C07D 491/048 (2006.01); C07D 513/04 (2006.01);
U.S. Cl.
CPC ...
C07D 487/04 (2013.01); C07D 471/04 (2013.01); C07D 487/16 (2013.01); C07D 491/048 (2013.01); C07D 513/04 (2013.01); C07D 519/00 (2013.01);
Abstract

Novel gyrase inhibitors and related compositions and methods are useful for impeding bacterial growth. Compounds of Formula I are disclosed:


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