The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.
The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.
Patent No.:
Date of Patent:
Sep. 20, 2016
Filed:
Dec. 18, 2013
Applicants:
Centre National DE LA Recherche Scientifique, Paris, FR;
Universite DE Reims Champagne-ardenne, Reims, FR;
Universite Paris Diderot Paris 7, Paris, FR;
Inventors:
Robert Dobb, Paris, FR;
Kevin Cariou, Paris, FR;
Stephanie Gourdain, Gif sur Yvette, FR;
Jean Maurice Delabar, Kremlin Bicetre, FR;
Nathalie Janel, Paris, FR;
Fernando Rodrigues Lima, Saint Maurice, FR;
Julien Dairou, Boulogne-Billancourt, FR;
Clement Denhez, Reims, FR;
Assignees:
Attorney:
Primary Examiner:
Int. Cl.
CPC ...
C07D 401/02 (2006.01); C07D 401/10 (2006.01); C07D 471/04 (2006.01);
U.S. Cl.
CPC ...
C07D 471/04 (2013.01);
Abstract
The present invention discloses compositions of novel DYRK1A protein inhibitors based on a 3,5-diarylazaindole motif and their preparation and use as medications in the treatment of cognitive disorders associated with dysfunction of DYRK1A protein, with Down's syndrome and with Alzheimer's disease.