The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Jul. 12, 2016

Filed:

Jul. 12, 2013
Applicant:

Khondrion Ip B.v., Beuningen Gld, NL;

Inventors:
Assignee:

Khondiron IP B.V., Beuningen, NL;

Attorneys:
Primary Examiner:
Int. Cl.
CPC ...
C07D 311/66 (2006.01); A61Q 19/08 (2006.01); C07D 413/12 (2006.01); A61K 8/49 (2006.01);
U.S. Cl.
CPC ...
C07D 311/66 (2013.01); A61K 8/498 (2013.01); A61Q 19/08 (2013.01); C07D 413/12 (2013.01); A61K 2800/74 (2013.01);
Abstract

The invention relates to novel compounds that are useful for modulating mitochondrial morphology and/or expression of OXPHOS enzymes and/or cellular ROS. The compounds are derivatives of TroloxrM wherein the carboxylic acid moiety is replaced by an amide moiety and wherein the nitrogen atom of the amide moiety is connected via a linker to a cationic nitrogen atom. The compounds of the invention are formulated into pharmaceutical or cosmetic compositions. The invention further relates to methods wherein the compounds of the invention are used for treating or preventing mitochondrial disorders, conditions associated with mitochondrial dysfunction, including adverse drug effects, and/or neoplastic diseases. The invention also relates to cosmetic methods for treating or delaying further aging of the skin and veterinary applications.


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