The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.
The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.
Patent No.:
Date of Patent:
May. 24, 2016
Filed:
Jan. 09, 2012
Applicants:
Markus Klein, Darmstadt, DE;
Christos Tsaklakidis, Weinheim, DE;
Hans Guehring, Eltville, DE;
Brigitta Leuthner, Darmstadt, DE;
Inventors:
Markus Klein, Darmstadt, DE;
Christos Tsaklakidis, Weinheim, DE;
Hans Guehring, Eltville, DE;
Brigitta Leuthner, Darmstadt, DE;
Assignee:
MERCK PATENT GMBH, Darmstadt, DE;
Primary Examiner:
Assistant Examiner:
Int. Cl.
CPC ...
C07K 5/10 (2006.01); A61K 38/08 (2006.01); C07K 5/02 (2006.01); A61K 38/06 (2006.01); A61K 38/07 (2006.01); A61K 45/06 (2006.01); C07K 5/087 (2006.01); C07K 5/103 (2006.01);
U.S. Cl.
CPC ...
A61K 38/08 (2013.01); A61K 38/06 (2013.01); A61K 38/07 (2013.01); A61K 45/06 (2013.01); C07K 5/0205 (2013.01); C07K 5/0812 (2013.01); C07K 5/101 (2013.01); C07K 5/1002 (2013.01);
Abstract
The present invention relates to compounds of the formula (I) and in particular medicaments comprising at least one compound of the formula (I) for use in the treatment and/or prophylaxis of physiological and/or pathophysiological states in the triggering of which cathepsin D is involved, in particular for use in the treatment and/or prophylaxis of arthrosis, traumatic cartilage injuries, arthritis, pain, allodynia or hyperalgesia.