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The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Patent No.:

US 9340500 B1

PDFFull Text
Expired
Date of Patent:
May. 17, 2016

Filed:

Apr. 18, 2012

Aromatic heterocyclic derivative having trpv4-inhibiting activity

Applicant:

Akira Yukimasa, Toyonaka, JP;

Inventor:

Akira Yukimasa, Toyonaka, JP;

Assignee:

SHIONOGI & CO., LTD., Osaka, JP;

Attorney:

Wenderoth, Lind & Ponack, L.L.P.

Primary Examiner:

Rebecca Anderson

Int. Cl.
CPC ...
C07D 403/12 (2006.01); C07D 403/04 (2006.01); C07D 401/04 (2006.01); C07D 409/12 (2006.01); C07D 405/12 (2006.01); C07D 413/04 (2006.01); C07D 417/12 (2006.01); C07D 417/14 (2006.01); C07D 207/34 (2006.01); C07D 213/82 (2006.01); C07D 231/14 (2006.01); C07D 233/90 (2006.01); C07D 401/12 (2006.01); C07D 209/08 (2006.01);
U.S. Cl.
CPC ...
C07D 207/34 (2013.01); C07D 209/08 (2013.01); C07D 213/82 (2013.01); C07D 231/14 (2013.01); C07D 233/90 (2013.01); C07D 401/04 (2013.01); C07D 401/12 (2013.01); C07D 403/04 (2013.01); C07D 403/12 (2013.01); C07D 405/12 (2013.01); C07D 409/12 (2013.01); C07D 413/04 (2013.01); C07D 417/12 (2013.01); C07D 417/14 (2013.01);
Abstract

A compound having TRPV4 inhibitory activity or a pharmaceutically acceptable salt thereof is provided. The present invention is related to a compound represented by the formula (I), wherein Ris substituted or unsubstituted alkyl or the like; Ris hydrogen or substituted or unsubstituted alkyl; Ris hydrogen, halogen, substituted or unsubstituted alkyl, substituted or unsubstituted cycloalkyl, substituted or unsubstituted nonaromatic heterocyclic group or the like; -L- is —C(=0)—NRor the like; X is substituted or unsubstituted aryl, substituted or unsubstituted heteroaryl or the like, or a pharmaceutically acceptable salt thereof.

Find Patent Forward Citations

Yukimasa, Akira. (2016). Aromatic heterocyclic derivative having trpv4-inhibiting activity (U.S. Patent No. 9340500). U.S. Patent and Trademark Office. https://idiyas.com/patent/badge/9340500

Data source: USPTO (United States Patent and Trademark Office) public patent records. Weekly synchronization. How IDiyas builds this profile

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