The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Patent No.:

US 9273049 B1

PDF
Full Text
Expired
Date of Patent:
Mar. 01, 2016

Filed:

Nov. 09, 2010
Applicants:

Wilna Liebenberg, Potchefstroom, ZA;

Nicole Stieger, Potchefstroom, ZA;

Inventors:

Wilna Liebenberg, Potchefstroom, ZA;

Nicole Stieger, Potchefstroom, ZA;

Assignee:
Attorney:
Primary Examiner:
Assistant Examiner:
Int. Cl.
CPC ...
A61K 9/00 (2006.01); C07D 471/14 (2006.01);
U.S. Cl.
CPC ...
C07D 471/14 (2013.01); Y10T 428/2982 (2015.01);
Abstract

The invention provides a method for increasing the solubility of nevirapine, including the steps of rendering nevirapine in a gaseous phase; and rendering the gaseous phase in a relatively more soluble solid particulate form. The invention further provides for a crystalline Form-VI () of nevirapine having an X-ray diffraction pattern of (2-theta values in degrees) 9.2953, 11.2023, 12.7019, 12.9796, 13.5273, 15.4670, 17.2597, 19.1038, 19.7267, 21.1303, 22.9381, 25.5589, 26.4913, 27.2150, 27.7283, 29.7134, and 33.8343 degrees two theta. The invention further provides for the preparation of microspherical and/or nanospherical Form-V () and crystalline Form-VI () of nevirapine as well as novel dosage forms including parenteral-, inhalant-, transdermal- and oral dosage forms.


Find Patent Forward Citations

Liebenberg, Wilna. (2016). Method for increasing the solubility of nevirapine (U.S. Patent No. 9273049). U.S. Patent and Trademark Office. https://idiyas.com/patent/badge/9273049

Data source: USPTO (United States Patent and Trademark Office) public patent records. Weekly synchronization. How IDiyas builds this profile

Loading…