The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.
The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.
Patent No.:
Date of Patent:
Feb. 02, 2016
Filed:
Nov. 21, 2011
Applicants:
Andreas Hafner, Gelterkinden, CH;
Fritz Blatter, Reinach, CH;
Martin Szelagiewicz, Basel, CH;
Bernd Siebenhaar, Kandern-Wollbach, DE;
Inventors:
Andreas Hafner, Gelterkinden, CH;
Fritz Blatter, Reinach, CH;
Martin Szelagiewicz, Basel, CH;
Bernd Siebenhaar, Kandern-Wollbach, DE;
Assignee:
BASF SE, Ludwigshafen, DE;
Primary Examiner:
Assistant Examiner:
Int. Cl.
CPC ...
C07D 239/42 (2006.01); C07C 29/00 (2006.01); C07C 31/26 (2006.01); A61K 31/505 (2006.01); A61K 47/26 (2006.01); A61K 47/48 (2006.01);
U.S. Cl.
CPC ...
C07D 239/42 (2013.01); C07C 29/00 (2013.01); C07C 31/26 (2013.01); A61K 31/505 (2013.01); A61K 47/26 (2013.01); A61K 47/4893 (2013.01);
Abstract
A novel solid form of Rosuvastatin comprises as the active ingredient a salt of bis[(E)-7-[4-(4-fluorophenyl)-6-isopropyl-2-[methyl(methylsulfonyl)-amino]pyrimidin-5-yl]-(3R,5S)-3,5-dihydroxyhept-6-enoic acid] and sorbitol. The crystal comprising the two components, and minor amounts of water, shows improved properties such as crystallization behavior and stability.