The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.
The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.
Patent No.:
Date of Patent:
Nov. 17, 2015
Filed:
Mar. 02, 2010
Michel Perez, Castres, FR;
Marie Lamothe, Castres, FR;
Didier Junquero, Castres, FR;
Yves Rival, Lagarrigue, FR;
Michel Perez, Castres, FR;
Marie Lamothe, Castres, FR;
Didier Junquero, Castres, FR;
Yves Rival, Lagarrigue, FR;
PIERRE FABRE MEDICAMENT, Boulogne-Billancourt, FR;
Abstract
The object of the present invention is benzothiazine derivatives having the capability of inhibiting 11β-HSD1 not only at an enzymatic level but also at a cell level. The compounds of the present invention are of general formula (I). Wherein notably Rrepresents a hydrogen or OR1 represents an ester or an ether. Rrepresents a naphthyl or a 1,2,3,4-tetrahydro-naphthalene or a biphenyl or phenyl pyridine or a substituted phenyl. Rrepresents a methyl or ethyl; Rand R'represent a hydrogen.