The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Nov. 03, 2015

Filed:

Feb. 23, 2015
Applicant:

Genzyme Corporation, Cambridge, MA (US);

Inventors:

John L. Kane, Jr., Stow, MA (US);

Gloria Matthews, Boylston, MA (US);

Markus Metz, Brookline, MA (US);

Michael Kothe, Medway, MA (US);

Jinyu Liu, Acton, MA (US);

Andrew Scholte, Somerville, MA (US);

Assignee:

GENZYME CORPORATION, Cambridge, MA (US);

Attorney:
Primary Examiner:
Int. Cl.
CPC ...
C07D 471/04 (2006.01); C07D 401/12 (2006.01); C07D 401/14 (2006.01); C07D 471/08 (2006.01); C07D 413/14 (2006.01); C07D 519/00 (2006.01); C07D 471/10 (2006.01); C07D 405/14 (2006.01); C07D 403/04 (2006.01); C07D 401/04 (2006.01); C07D 413/04 (2006.01);
U.S. Cl.
CPC ...
C07D 471/04 (2013.01); C07D 401/04 (2013.01); C07D 401/12 (2013.01); C07D 401/14 (2013.01); C07D 403/04 (2013.01); C07D 405/14 (2013.01); C07D 413/04 (2013.01); C07D 413/14 (2013.01); C07D 471/08 (2013.01); C07D 471/10 (2013.01); C07D 519/00 (2013.01);
Abstract

Tropomyosin-related kinase inhibitors (Trk inhibitors) are small molecule compounds useful in the treatment of disease. Trk inhibitors can be used as pharmaceutical agents and in pharmaceutical compositions. Trk inhibitors are useful in the treatment of inflammatory diseases, autoimmune disease, defects of bone metabolism and/or cancer, and are particularly useful in the treatment of osteoarthritis (OA), pain, and pain associated with OA. Trk inhibitors are also useful for inhibiting tropomyosin-related kinase A (TrkA), tropomyosin-related kinase B (TrkB), tropomyosin-related kinase C (TrkC), and/or c-FMS (the cellular receptor for colony stimulating factor-1 (CSF-1)).


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