The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Nov. 03, 2015

Filed:

Oct. 05, 2009
Applicants:

Simon Green, Dundee, GB;

Sheelagh Frame, Dundee, GB;

Ian Fleming, Angus, GB;

Inventors:

Simon Green, Dundee, GB;

Sheelagh Frame, Dundee, GB;

Ian Fleming, Angus, GB;

Assignee:

Cyclacel Limited, London, GB;

Attorneys:
Primary Examiner:
Int. Cl.
CPC ...
C07D 473/34 (2006.01); A61K 31/52 (2006.01); A61K 45/06 (2006.01); A61K 31/517 (2006.01);
U.S. Cl.
CPC ...
A61K 45/06 (2013.01); A61K 31/517 (2013.01); A61K 31/52 (2013.01);
Abstract

The present invention relates to combination comprising (i) an ErbB inhibitor; and (ii) a CDK inhibitor, or a pharmaceutically acceptable salt thereof, selected from: (a) roscovitine; (b) 3-{9-isopropyl-6-[(pyridin-3-ylmethyl)-amino]-9H-purin-2-ylamino}-2-methyl-pentan-2-ol; (c) 3-{9-isopropyl-6-[(pyridin-3-ylmethyl)-amino]-9H-purin-2-ylamino}-pentan-2-ol; and (d) (2R,3S-3-(6-((4,6-dimethylpyridin-3-ylmethylamino)-9-isopropyl-9H-purin-2-ylamino)pentan-2-ol. Further aspects of the invention relate to pharmaceutical products and pharmaceutical compositions comprising combinations according to the invention, and methods of treatment using the same.


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