The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Patent No.:

US 9169232 B1

PDF
Full Text
Expired
Date of Patent:
Oct. 27, 2015

Filed:

Sep. 14, 2012
Applicants:

Sanjay Sukumar Saralaya, Bangalore, IN;

Akshaya Kunjyannaya, Bangalore, IN;

Shashiprabha, Bangalore, IN;

Shridhara Kanakamajalu, Bangalore, IN;

Kothapalli Sundarraja Rao, Bangalore, IN;

Kuppuswamy Nagarajan, Bangalore, IN;

Inventors:

Sanjay Sukumar Saralaya, Bangalore, IN;

Akshaya Kunjyannaya, Bangalore, IN;

Shashiprabha, Bangalore, IN;

Shridhara Kanakamajalu, Bangalore, IN;

Kothapalli Sundarraja Rao, Bangalore, IN;

Kuppuswamy Nagarajan, Bangalore, IN;

Assignee:
Attorneys:
Primary Examiner:
Int. Cl.
CPC ...
C07D 317/36 (2006.01); C07D 317/40 (2006.01);
U.S. Cl.
CPC ...
C07D 317/36 (2013.01); C07D 317/40 (2013.01);
Abstract

The present invention relates to atovaquone prodrug compound of formula (I). Accordingly, present invention provides a process involving condensation of Atovaquone (II) with 5-methyl-4-chloromethyl dioxalone (III) in suitable solvent system and optionally followed by distillation and crystallization to provide Atovaquone prodrug compound of formula (I) in high yields, purity, and suitable for large-scale manufacture.


Find Patent Forward Citations

Saralaya, Sanjay. (2015). 3-(5-methyl-2-oxo-l, 3-dioxol-4-yl) methyloxy-2-trans-[(4-chloro phenyl) cyclohexyl][1,4]naphthaquinone-atovaquone prodrug (U.S. Patent No. 9169232). U.S. Patent and Trademark Office. https://idiyas.com/patent/badge/9169232

Data source: USPTO (United States Patent and Trademark Office) public patent records. Weekly synchronization. How IDiyas builds this profile

Loading…