The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Oct. 20, 2015

Filed:

Sep. 24, 2010
Applicants:

Robert A. Mitchell, Louisville, KY (US);

John O. Trent, Louisville, KY (US);

Pooran Chand, Birmingham, AL (US);

Gilles Hugues Tapolsky, Louisville, KY (US);

Inventors:

Robert A. Mitchell, Louisville, KY (US);

John O. Trent, Louisville, KY (US);

Pooran Chand, Birmingham, AL (US);

Gilles Hugues Tapolsky, Louisville, KY (US);

Assignees:
Attorney:
Primary Examiner:
Assistant Examiner:
Int. Cl.
CPC ...
C07D 239/02 (2006.01); A01N 43/54 (2006.01); A61K 31/505 (2006.01); C07D 239/30 (2006.01); C07D 239/38 (2006.01); C07D 239/42 (2006.01); C07D 401/04 (2006.01); C07D 405/04 (2006.01); C07D 409/04 (2006.01);
U.S. Cl.
CPC ...
C07D 239/30 (2013.01); C07D 239/38 (2013.01); C07D 239/42 (2013.01); C07D 401/04 (2013.01); C07D 405/04 (2013.01); C07D 409/04 (2013.01);
Abstract

Compounds useful for the inhibition of macrophage migration inhibitory factor (MIF) are provided herein, having the Formula (I): wherein A is selected from the group consisting of aromatic or non-aromatic rings, bicyclic rings, polycyclic rings, alkenes or alkynes; B is H, OH, OR, SR, NH2, NHR, or alkyl; R is H or alkyl, and X and Y are independently N or CH, but one of X and Y must be N. Also provided are pharmaceutical compositions comprising a Formula I compound and methods for the treatment of MIF-implicated diseases or conditions, comprising administering a safe and effective amount of a Formula I compound.


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