The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Oct. 20, 2015

Filed:

May. 16, 2012
Applicants:

Rasmus Irming Jølck, Valby, DK;

Jonas Rosager Henriksen, Allerød, DK;

Torben Gjetting, Jyllinge, DK;

Thomas Lars Andresen, Vanløse, DK;

Inventors:

Rasmus Irming Jølck, Valby, DK;

Jonas Rosager Henriksen, Allerød, DK;

Torben Gjetting, Jyllinge, DK;

Thomas Lars Andresen, Vanløse, DK;

Assignee:
Attorney:
Primary Examiner:
Int. Cl.
CPC ...
A61K 47/48 (2006.01); A61K 31/282 (2006.01); A61K 31/7088 (2006.01); A61K 9/127 (2006.01); A61K 9/14 (2006.01);
U.S. Cl.
CPC ...
A61K 47/48838 (2013.01); A61K 9/1272 (2013.01); A61K 9/145 (2013.01); A61K 31/282 (2013.01); A61K 31/7088 (2013.01); A61K 47/48053 (2013.01); A61K 47/48215 (2013.01); A61K 47/48238 (2013.01); A61K 47/48323 (2013.01); A61K 47/48338 (2013.01); A61K 47/48815 (2013.01); A61K 47/48853 (2013.01); Y10S 977/80 (2013.01); Y10S 977/801 (2013.01); Y10S 977/907 (2013.01);
Abstract

The present application discloses a nanoparticle comprising compounds of the formula A-B-C(-D), wherein A designates an anchoring moiety having self-organizing properties in relation to the nanoparticle; B designates a cleavable linker; C designates an anionic moiety having a net charge of at least −2 at pH 6.0; and D, which is optional, designates a polymer moiety which induces long circulating properties of the nanoparticle in mammalian tissue; and wherein the average net charge of the compounds is at least −1 at pH 6.0. The application also discloses the individual compounds of the formula A-B-C(-D) as well as a drug delivery system comprising the self-organized nanoparticle having included in the interior thereof one or more pharmaceutically active agents and/or diagnostically relevant species, and a method of treating a cancerous or inflammatory condition in a mammal, involving the administration of the drug delivery system to the mammal.


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