The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Jun. 23, 2015

Filed:

Apr. 18, 2013
Applicant:

Changzhou Le Sun Pharmaceuticals Limited, Jiangsu, CN;

Inventors:

Shudong Wang, Adelaide, AU;

Hao Shao, Nottingham, GB;

Assignee:
Attorney:
Primary Examiner:
Int. Cl.
CPC ...
C07D 401/00 (2006.01); C07D 417/04 (2006.01);
U.S. Cl.
CPC ...
C07D 417/04 (2013.01);
Abstract

The present invention relates to compounds of formula (I): wherein Ris NHor NHMe; Ris halo; and one of Ror Ris hydrogen and the other is selected from —SONH, —SONHMe or —SONMe, —SONHEt, or —SONEt; or a pharmaceutically acceptable salt or solvate thereof. The compounds of formula (I) are inhibitors of protein kinases, especially cyclic dependent kinases (CDKs) such as CDK9. The present invention also relates to processes for the preparation of these compounds, to pharmaceutical compositions comprising them, and to their use in the treatment of proliferative disorders, such as cancer, as well as other diseases or conditions in which protein kinase/CDK activity is implicated.


Find Patent Forward Citations

Wang, Shudong. (2015). Therapeutic compounds (U.S. Patent No. 9062039). U.S. Patent and Trademark Office. https://idiyas.com/patent/badge/9062039

Data source: USPTO (United States Patent and Trademark Office) public patent records. Weekly synchronization. How IDiyas builds this profile

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