The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.
The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.
Patent No.:
Date of Patent:
Jun. 02, 2015
Filed:
Sep. 06, 2013
Applicant:
Gilead Sciences, Inc., Foster City, CA (US);
Inventors:
Jeff A. Zablocki, Mountain View, CA (US);
Elfatih O. Elzein, Fremont, CA (US);
Venkata P. Palle, Pune, IN;
Luiz Belardinelli, Palo Alto, CA (US);
Assignee:
Gilead Sciences, Inc., Foster City, CA (US);
Primary Examiner:
Int. Cl.
CPC ...
A61K 31/70 (2006.01); C07H 19/167 (2006.01); C07H 19/173 (2006.01); A01N 43/04 (2006.01); C07H 19/16 (2006.01); C07D 473/34 (2006.01);
U.S. Cl.
CPC ...
C07H 19/16 (2013.01); C07D 473/34 (2013.01);
Abstract
The present disclosure provides a process for the preparation of 2-adenosine N-pyrazole compounds exemplified by the structure shown below that are potent and selective agonists for Aadenosine receptor, compositions comprising these compounds, and methods for using these compound to stimulate mammalian coronary vasodilatation for imaging the heart.