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The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Patent No.:

US 9045445 B1

PDFFull Text
Date of Patent:
Jun. 02, 2015

Filed:

Jun. 02, 2011

Glycine transporter-1 inhibitors, methods of making them, and uses thereof

Applicants:

Christopher L. Cioffi, Troy, NY (US);

Mark A. Wolf, Denlanson, NY (US);

Peter R. Guzzo, Niskayuna, NY (US);

Shuang Liu, Schenectady, NY (US);

Kashinath Sadalapure, Singapore, SG;

Inventors:

Christopher L. Cioffi, Troy, NY (US);

Mark A. Wolf, Denlanson, NY (US);

Peter R. Guzzo, Niskayuna, NY (US);

Shuang Liu, Schenectady, NY (US);

Kashinath Sadalapure, Singapore, SG;

Assignee:

Albany Molecular Research, Inc., Albany, NY (US);

Attorney:

LeClairRyan, a Professional Corporation

Primary Examiner:

Golam M M Shameem

Int. Cl.
CPC ...
A61K 31/496 (2006.01); C07D 403/12 (2006.01); C07D 295/26 (2006.01); C07D 205/04 (2006.01); C07D 207/48 (2006.01); C07D 211/58 (2006.01); C07D 213/71 (2006.01); C07D 233/84 (2006.01); C07D 241/04 (2006.01); C07D 249/04 (2006.01); C07D 309/14 (2006.01); C07D 313/04 (2006.01); C07D 405/12 (2006.01); C07D 487/08 (2006.01);
U.S. Cl.
CPC ...
C07D 295/26 (2013.01); C07D 205/04 (2013.01); C07D 207/48 (2013.01); C07D 211/58 (2013.01); C07D 213/71 (2013.01); C07D 233/84 (2013.01); C07D 241/04 (2013.01); C07D 249/04 (2013.01); C07D 309/14 (2013.01); C07D 313/04 (2013.01); C07D 405/12 (2013.01); C07D 487/08 (2013.01);
Abstract

The compounds of the present invention are represented by the following formula (I): wherein the substituents R, R, R, R, (R), R, A, X, and Y are as defined herein. The compounds are useful in methods of treating a disorder which is created by or is dependent upon inhibiting GlyT-1.

Find Patent Forward Citations

Cioffi, Christopher. (2015). Glycine transporter-1 inhibitors, methods of making them, and uses thereof (U.S. Patent No. 9045445). U.S. Patent and Trademark Office. https://idiyas.com/patent/badge/9045445

Data source: USPTO (United States Patent and Trademark Office) public patent records. Weekly synchronization. How IDiyas builds this profile

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