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The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Patent No.:

US 9029387 B1

PDFFull Text
Expired
Date of Patent:
May. 12, 2015

Filed:

Feb. 28, 2011

Benzonaphthyridinamines as autotaxin inhibitors

Applicants:

Wolfgang Staehle, Ingelheim, DE;

Melanie Schultz, Darmstadt, DE;

Kai Schiemann, Seeheim-Jugenheim, DE;

Inventors:

Wolfgang Staehle, Ingelheim, DE;

Melanie Schultz, Darmstadt, DE;

Kai Schiemann, Seeheim-Jugenheim, DE;

Assignee:

Merck Patent GmbH, Darmstadt, DE;

Attorney:

Millen, White, Zelano & Branigan, P.C.

Primary Examiner:

Samira Jean-Louis

Int. Cl.
CPC ...
A01N 43/42 (2006.01); A61K 31/44 (2006.01); A61K 31/497 (2006.01); A61K 31/535 (2006.01); C07D 471/00 (2006.01); C07D 491/00 (2006.01); C07D 498/00 (2006.01); C07D 513/00 (2006.01); C07D 515/00 (2006.01); C07D 401/00 (2006.01); C07D 413/00 (2006.01); C07D 471/04 (2006.01);
U.S. Cl.
CPC ...
C07D 471/04 (2013.01);
Abstract

The present invention relates to benzonaphthyridinamines of the formula (I) as autotaxin inhibitors and to the use thereof in the treatment and/or prophylaxis of physiological and/or pathophysiological conditions in which the inhibition, regulation and/or modulation of phosphodiesterase or lysophospholipase autotaxin plays a role, in particular of various types of cancer and autoimmune and inflammatory diseases.

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Staehle, Wolfgang. (2015). Benzonaphthyridinamines as autotaxin inhibitors (U.S. Patent No. 9029387). U.S. Patent and Trademark Office. https://idiyas.com/patent/badge/9029387

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