The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Apr. 21, 2015

Filed:

Jun. 08, 2012
Applicants:

Yoshiro Niitsu, Hokkaido, JP;

Victor Knopov, Oceanside, CA (US);

Joseph E. Payne, Oceanside, CA (US);

Zheng Hou, San Diego, CA (US);

John A. Gaudette, Poway, CA (US);

Violetta Akopian, Oceanside, CA (US);

Richard P. Witte, San Diego, CA (US);

Mohammad Ahmadian, Carlsbad, CA (US);

Loren A. Perelman, San Diego, CA (US);

Yasunobu Tanaka, Osaka, JP;

Priya Karmali, San Diego, CA (US);

Sridhar C. Nagarajan, San Diego, CA (US);

Inventors:

Yoshiro Niitsu, Hokkaido, JP;

Victor Knopov, Oceanside, CA (US);

Joseph E. Payne, Oceanside, CA (US);

Zheng Hou, San Diego, CA (US);

John A. Gaudette, Poway, CA (US);

Violetta Akopian, Oceanside, CA (US);

Richard P. Witte, San Diego, CA (US);

Mohammad Ahmadian, Carlsbad, CA (US);

Loren A. Perelman, San Diego, CA (US);

Yasunobu Tanaka, Osaka, JP;

Priya Karmali, San Diego, CA (US);

Sridhar C. Nagarajan, San Diego, CA (US);

Assignee:
Attorney:
Primary Examiner:
Assistant Examiner:
Int. Cl.
CPC ...
A61K 31/225 (2006.01); C07C 69/34 (2006.01); A61K 9/127 (2006.01); A61K 31/7052 (2006.01); A61K 47/18 (2006.01); A61K 9/00 (2006.01); A61K 9/10 (2006.01); A61K 31/713 (2006.01); C12N 15/113 (2010.01);
U.S. Cl.
CPC ...
A61K 47/186 (2013.01); A61K 9/0019 (2013.01); A61K 9/10 (2013.01); A61K 9/1271 (2013.01); A61K 31/713 (2013.01); C12N 15/113 (2013.01);
Abstract

Here described are compounds of formula I: wherein Rand Ris independently selected from a group consisting of Cto Calkyl, Cto Calkenyl, and oleyl group; wherein Rand Rare independently selected from a group consisting of Cto Calkyl, and Cto Calkanol; wherein X is selected from a group consisting of —CH—, —S—, and —O— or absent; wherein Y is selected from —(CH), —S(CH), —O(CH)—, thiophene, —SO(CH)—, and ester, wherein n=1-4; wherein a=1-4; wherein b=1-4; wherein c=1-4; and wherein Z is a counterion; as well as compositions and pharmaceutical formulations including compounds of formula I which are useful for the delivery of therapeutic agents; and methods of using these compositions and formulations.


Find Patent Forward Citations

Loading…